STRUCTURAL BIOLOGY & CHEMICAL EVIDENCEDataset v1.2 · Phase 6D · Comparative experimental recognition environments

small molecule preparation

compound 7 (Collie 2025)

Published observations for this preparation and the reported assay constructs.

exact single CCD identity

Identity scope

Measured preparation

Preparation ID
PREP:COLLIE2025_7
Exact CCD identity
A1IEF
Modeled candidate components
None

Assay evidence

Published observations

4 records
Assay recordTarget and constructEndpointReported resultSource
PWWP:ASSAY:0017NSD2 PWWP1
Construct 208–368
SPR Kd= 0.15 µM ± 0.02
SD
PMID:40959233
Conditions and interpretation
PWWP:ASSAY:0024NSD2 PWWP1
Construct 211–350
SPR Kd= 0.76 µM ± 0.01
SD
PMID:40959233
Conditions and interpretation
PWWP:ASSAY:0029NSD2 PWWP1
Construct 208–368
HTRF displacement IC50= 0.21 µM ± 0.01
SEM
PMID:40959233
Conditions and interpretation
PWWP11:ASSAY:0004NSD3 PWWP1
Construct 263–398
SPR Kd counter-screen> 30.0 µMPMID:40959233
Conditions and interpretation