STRUCTURAL BIOLOGY & CHEMICAL EVIDENCEDataset v1.2 · Phase 6D · Comparative experimental recognition environments

small molecule preparation

compound 5 (Collie 2025)

Published observations for this preparation and the reported assay constructs.

assayed stereoisomeric mixture not single chemical identity

Identity scope

Measured preparation

Preparation ID
PREP:COLLIE2025_5
Exact CCD identity
Unresolved at exact-identity level
Modeled candidate components
None

Assay evidence

Published observations

3 records
Assay recordTarget and constructEndpointReported resultSource
PWWP:ASSAY:0015NSD2 PWWP1
Construct 208–368
SPR Kd= 0.16 µM ± 0.03
SD
PMID:40959233
Conditions and interpretation
PWWP:ASSAY:0022NSD2 PWWP1
Construct 211–350
SPR Kd= 0.92 µM ± 0.03
SD
PMID:40959233
Conditions and interpretation
PWWP11:ASSAY:0002NSD3 PWWP1
Construct 263–398
SPR Kd counter-screen> 30.0 µMPMID:40959233
Conditions and interpretation